Award details

De novo design of novel emulsifiers based on a protein scaffold for use in polymeric encapsulation of macromolecules

ReferenceE19380
Principal Investigator / Supervisor Dr Christopher van der Walle
Co-Investigators /
Co-Supervisors
Institution University of Strathclyde
DepartmentInst of Pharmacy and Biomedical Sci
Funding typeResearch
Value (£) 131,868
StatusCompleted
TypeResearch Grant
Start date 01/02/2004
End date 30/04/2006
Duration27 months

Abstract

A major obstacle for encapsulation of therapeutic proteins in polylactide-co-glycolide (PLGA) microspheres remains the emulsion phase which causes protein denaturation and loss of activity. The current use of additives and synthetic emulsifiers is not ideal and, surprisingly, protein emulsifiers have been largely ignored. This speculative proposal intends to explore their potential by building on the current understanding of characteristics typical of protein emulsifiers. Structure-prediction will be used to superpose these characteristics onto a human protein scaffold with minimal mutation. Mutants will be expressed and tested, allowing quantification of the resultant emulsifying activity with respect to the structural-parameters used.

Summary

unavailable
Committee Closed Committee - Engineering & Biological Systems (EBS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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