Award details

Mechanisms kinetics of membrane transport and structure-activity relationships of membrane translocating peptides

ReferenceE14784
Principal Investigator / Supervisor Professor Anthony Smith
Co-Investigators /
Co-Supervisors
Institution University of Bath
DepartmentPharmacy and Pharmacology
Funding typeResearch
Value (£) 166,994
StatusCompleted
TypeResearch Grant
Start date 01/12/2000
End date 31/05/2004
Duration42 months

Abstract

Membrane translocating peptides (MTP) appear to cross biological membranes by passive processes and can be used to deliver active polypeptides to intracellular locations. This project will investigate the mechanisms of action of known MTPs, and quantify the kinetics of mass transport at the cellular and tissue level. Emphasis will be placed on determining the common structural requirements for translocation of existing MTPs, and examining the effects of polypeptide payloads on transport kinetics. Structure-activity studies will be carried out using a random mutagenesis strategy, with a view to designing optimal features of MTPs. The project will provide a fundamental evaluation of MTPs for delivery of therapeutic peptides.

Summary

unavailable
Committee Closed Committee - Engineering & Biological Systems (EBS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
terms and conditions of use (opens in new window)
export PDF file