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Synthesis and applications of porphocyanine-oligodeoxynucleotide conjugates as photoactive antisense agents

ReferenceE12509
Principal Investigator / Supervisor Professor Ross Boyle
Co-Investigators /
Co-Supervisors
Dr Julie Lloyd, Dr Minnie O'Farrell
Institution University of Hull
DepartmentChemistry
Funding typeResearch
Value (£) 172,220
StatusCompleted
TypeResearch Grant
Start date 01/10/2000
End date 24/05/2004
Duration43 months

Abstract

Conjugates of porphocyanine, a novel class of expanded porphyrin, and oligodeoxynucleotides will be synthesised and assayed for potential as photoactive antisense agents. Conjugates of porphocyanine and oligodeoxynucleotides will be investigated using a rapid screening system based on inhibition of a reporter gene which expresses beta- galactosidase. Promising conjugates will then be assayed for their ability to specifically inhibit human oncogene expression in cells expressing normal and mutant human ras p21. Fluorescence microscopy will be used to study uptake and intracellular distribution of conjugates; substituents on the porphocyanine will be modified to optimise these factors.

Summary

unavailable
Committee Closed Committee - Engineering & Biological Systems (EBS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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