Award details

Development of an enzyme-catalysed desymmetrisation of prochiral ketones

ReferenceE09803
Principal Investigator / Supervisor Dr Andrew Carnell
Co-Investigators /
Co-Supervisors
Institution University of Liverpool
DepartmentChemistry
Funding typeResearch
Value (£) 179,437
StatusCompleted
TypeResearch Grant
Start date 20/07/1998
End date 20/07/2001
Duration36 months

Abstract

We wish to develop a novel biotransformation which uses readily available hydrolytic enzymes for the production of chiral enol esters from a symmetrical cyclic and bicyclic ketones. These enol esters are extremely useful for the synthesis of fine chemicals and pharmaceuticals. We have demonstrated the success (Tet Lett. 1997, 38, 7781) of this approach with the model compound 4-cyano-4- phenylcyclohexanone. We propose to establish optimum conditions for four classes of substrate, demonstrate the synthetic potential of the chiral enol esters and show that the process is amenable to scale up.

Summary

unavailable
Committee Closed Committee - Engineering & Biological Systems (EBS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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