Award details

Molecular mechanisms of gating of G-protein- activated inwardly rectifying K channels

ReferenceC09333
Principal Investigator / Supervisor Dr Ruth Murrell-Lagnado
Co-Investigators /
Co-Supervisors
Institution University of Cambridge
DepartmentPharmacology
Funding typeResearch
Value (£) 179,304
StatusCompleted
TypeResearch Grant
Start date 17/08/1998
End date 31/12/2001
Duration40 months

Abstract

G protein-activated inward rectifier K+ channels (GIRKs) are found in central neurones where they act to suppress firing. They couple to receptors via pertussis toxin-sensitive G-proteins and are directly activated by the binding of G beta g subunits. They have been cloned and shown to have 2 transmembrane regions. The native neuronal channels are heteromers composed of GIRK1 and GIRK2. We have made a series of chimeric subunits composed of GIRK1 and GIRK2 and these differ in their voltage-dependent gating properties and also in their gating by internal ligands. The aim of this proposal is to understand the molecular mechanisms of gating of recombinant GIRKs expressed in Xenopus oocytes using electrophysiological and molecular biological methods.

Summary

unavailable
Committee Closed Committee - Biochemistry & Cell Biology (BCB)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
terms and conditions of use (opens in new window)
export PDF file