Award details

Energy coupling and the basis of specificity of Escherichia coli topoisomerase IV

ReferenceC06672
Principal Investigator / Supervisor Dr Andrew Bates
Co-Investigators /
Co-Supervisors
Institution University of Liverpool
DepartmentSch of Biological Sciences
Funding typeResearch
Value (£) 155,201
StatusCompleted
TypeResearch Grant
Start date 01/03/1997
End date 01/03/2000
Duration36 months

Abstract

In recent years, topoisomerase IV, a new bacterial type II topoisomerase and antibacterial drug target has been identified, which is specifically involved in the ATP-dependent decatenation (unlinking) of daughter chromosomes. It is proposed to investigate the detailed biochemistry of E. coli topo IV, with a view to the elucidation of the basis of the selective coupling of ATP hydrolysis to the decatenation reaction, using assays of ATPase activity, ADPNP-dependent reactions and quinolone drug inhibition, with DNA substrates designed to reveal relaxation or decatenation activity. The structural basis of the enzyme's specificity will be addressed by characterisation of mutant and engineered forms of the enzyme.

Summary

unavailable
Committee Closed Committee - Biochemistry & Cell Biology (BCB)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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