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Mechanism of CMP-Neu5Ac hydroxylase

ReferenceBCI06184
Principal Investigator / Supervisor Professor Timothy Bugg
Co-Investigators /
Co-Supervisors
Institution University of Southampton
DepartmentSch of Chemistry
Funding typeResearch
Value (£) 42,159
StatusCompleted
TypeResearch Grant
Start date 17/01/1997
End date 17/02/1998
Duration13 months

Abstract

The objectives of the proposed research are to elucidate the stereochemistry and mechanism of CMP-N-acetylneuraminic acid hydroxylase, a non-haem iron (II) dependent oxygenase enzyme involved in the biosynthesis of sialic acid-containing glycoconjugates. A series of N-acyl-neuraminic acid analogues will be synthesised from D-glycosamine using the enzyme N-acetylneuraminic acid aldolase. The stereochemistry of the enzymatic reaction will be deduced using stereospecifically labelled N-propionyl-analogues, and the intermediacy of enolate vs. radical intermediates will be assessed using isotope exchange and cyclopropyl radical traps.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative Biological Chemistry Initiative (BCI) [1995]
Funding SchemeX – not Funded via a specific Funding Scheme
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