Award details

Novel inhibitors as probes for the molecular biology of O-glycosylated proteins

ReferenceB19303
Principal Investigator / Supervisor Professor Timothy Gallagher
Co-Investigators /
Co-Supervisors
Dr Anthony Corfield
Institution University of Bristol
DepartmentChemistry
Funding typeResearch
Value (£) 298,424
StatusCompleted
TypeResearch Grant
Start date 01/12/2003
End date 31/03/2007
Duration40 months

Abstract

O-Glycosylated proteins are responsible for essential cell functions and at mucosal surfaces for the innate barrier protection against the external environment. They are formed through well- characterised pathways in all cells and are defective in colorectal cancer. Selective manipulation of these processes will advance significantly our knowledge of their overall importance to the normal cell and facilitate intervention in defined disease aberrations. Inhibition of these pathways has been achieved using O-benzyl GalNAc but no other compounds have been tested. The synthesis of a family of novel analogues will enable selective manipulation of biologically critical O-glycosylation pathways to be achieved.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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