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Molecular basis of PP2A regulation through methylation-dependent assembly of heterotrimers

ReferenceB18126
Principal Investigator / Supervisor Professor Snezana Djordjevic
Co-Investigators /
Co-Supervisors
Institution University College London
DepartmentStructural Molecular Biology
Funding typeResearch
Value (£) 175,564
StatusCompleted
TypeResearch Grant
Start date 15/02/2003
End date 15/02/2006
Duration36 months

Abstract

Protein phosphataste 2A is a ubiquitous enzyme with a range of diverse substrates. Substrate specificity and subcellular localisation is determined by more than 20 different regulatory subunits. Binding of regulatory subunits and heterotrimeric formation is dependent on carboxymethylation of the conserved terminal leucine residue of the catalytic subunit. This covalent modification is catalysed by the specific S-adenosylmethinine dependent methyltransferase while the reverse reaction of methylester hydrolysis is carried out by the unique methylesterase. How the two methylation enzymes are regulated is not known. The object of this proposal is to establish the molecular basis of the mechanisms of heterotrimeric assembly by investigating the three-dimensional structures of the methylation enzymes and their respective complexes with the catalytic subunit of PP2A.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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