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Study of the mechanism of pyrrole polymerisation with human mutant enzymes that accumulate stable catalytic intermediates

ReferenceB17399
Principal Investigator / Supervisor Professor Peter Shoolingin-Jordan
Co-Investigators /
Co-Supervisors
Institution University of Southampton
DepartmentCentre for Biological Sciences
Funding typeResearch
Value (£) 186,213
StatusCompleted
TypeResearch Grant
Start date 01/07/2002
End date 31/12/2005
Duration42 months

Abstract

The mechanism by which the pyrrole, porphobilinogen, is polymerised enzymically to give preuroporphyrinogen, the tetrapyrrole intermediate of haem synthesis, will be investigated using two naturally occurring human mutants of porphobilinogen deaminase that are defective in the chain extension mechanism. The mutants will be isolated as their stable mono, di, tri and tetrapyrrole enzyme-intermediate complexes and the individual X-ray structures will be solved. The structures will reveal the precise detail of the stepwise mechanism of tetrapyrrole chain synthesis. Other naturally occurring human mutants will be employed to investigate the assembly of the novel dipyrromethane cofactor that acts as the primer for tetrapyrrole chain synthesis.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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