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A computational investigation of G-protein coupled receptor dimerisation

ReferenceB17252
Principal Investigator / Supervisor Professor Christopher Reynolds
Co-Investigators /
Co-Supervisors
Institution University of Essex
DepartmentBiological Sciences
Funding typeResearch
Value (£) 128,100
StatusCompleted
TypeResearch Grant
Start date 01/03/2003
End date 28/02/2005
Duration24 months

Abstract

GPCR dimerization and heterodimerization and highly significant phenomena in signal transduction that have wide-ranging implications for many areas of research, particularly in the pharmaceutical industry. Despite a high level of international activity, including a small but highly significant UK contribution, the significance of GPCR dimerization for activity is not understood at the molecular level. Here we propose to investigate GPCR dimerization at the molecular level through a range of computational activities including bioinformatics and simulation. These studies will draw heavily on very recent biophysical, mutational and drug-binding data that permit key studies on the nature of the active receptor, the nature of the dimer and insig.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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