Award details

Achieving photo-control of protein activity: application to bZIP and bHLH DNA binding proteins

ReferenceB16000
Principal Investigator / Supervisor Professor Rudolf Allemann
Co-Investigators /
Co-Supervisors
Institution University of Birmingham
DepartmentSchool of Chemistry
Funding typeResearch
Value (£) 194,180
StatusCompleted
TypeResearch Grant
Start date 01/12/2001
End date 31/05/2005
Duration42 months

Abstract

The award holders have successfully designed, synthesised and characterised a peptide containing a photo- isomerisable cross-linker. Photo-isomerisation of the cross-linker leads to a change in the peptide conformation from random coil to alpha-helical. This work has already been extended to control the helicity of the leucine zipper peptide from GCNA4 (GCNA-ZIP), allowing photo-control of dimerization. We seek to extend this technology by application to two DNA binding proteins. The lessons already learnt on GCN4-ZIP will be used to produce a photo-controlled variant of the longer DNA-binding GCN4-bZIP. A different way of controlling activity will be tested by the direct control of the helicity of the basic (DNA binding) helix of MyoD, a BHLH protein.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
terms and conditions of use (opens in new window)
export PDF file