Award details

Crystallographic analysis of ligand binding to human serum albumin (HSA)

ReferenceB12706
Principal Investigator / Supervisor Professor Stephen Curry
Co-Investigators /
Co-Supervisors
Institution Imperial College London
DepartmentBiological Sciences
Funding typeResearch
Value (£) 181,328
StatusCompleted
TypeResearch Grant
Start date 20/03/2000
End date 17/07/2003
Duration40 months

Abstract

Human serum albumin (HSA) is an important plasma protein that binds fatty acids, a wide range of drugs and surface proteins of certain pathogenic bacteria. The interactions of HSA with its various ligands have been studied for many years, but there remains a dearth of structural information. Recently we published the first structure of HSA bound to fatty acid, its primary ligand. We now wish to extend our crystallographic structural analysis of HSA to incorporate (1) additional fatty acids (both saturated and unsaturated); (2) a range of drug compounds known to bind to the two primary drug binding sites on the protein (3) the GA- type albumin binding domain from bacterial surface proteins. This study should provide a wealth of new information on structural aspects of ligand binding to HSA.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
terms and conditions of use (opens in new window)
export PDF file