Award details

Resin screening and combinatorial fishing - a method of ligand self selection

ReferenceB09914
Principal Investigator / Supervisor Professor Mark Bradley
Co-Investigators /
Co-Supervisors
Institution University of Southampton
DepartmentSch of Chemistry
Funding typeResearch
Value (£) 149,884
StatusCompleted
TypeResearch Grant
Start date 11/11/1998
End date 11/01/2002
Duration38 months

Abstract

A method of unrivalled power in terms of compound number and ease of analysis will be developed for the combinatorial area. The aim is to enhance the numbers of compounds that can be screened in a library by several orders of magnitude but at the same time actually reduce the numbers of compounds that need to be synthesised. The modus operandi will be the dynamic generation of diversity and of enzyme self- selection strategy using a combination of solid and solution phase libraries and will use a 'resin capture strategy'. The process will enable multiple site binding and cooperativity to be investigated and exploited.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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