Award details

X-ray structural studies of saponin-detoxifying enzymes as targets for antifungal design

ReferenceB09174
Principal Investigator / Supervisor Professor Andrew Hemmings
Co-Investigators /
Co-Supervisors
Institution University of East Anglia
DepartmentBiological Sciences
Funding typeResearch
Value (£) 103,966
StatusCompleted
TypeResearch Grant
Start date 01/07/1998
End date 01/07/2000
Duration24 months

Abstract

Saponins are plant secondary metabolites with potent antifungal properties. A number of fungi can breach this defence by producing extracellular saponin-detoxifying enzymes. We wish to structurally characterise these enzymes and their mode of substrate binding as they constitute attractive targets for the design of specific antifungal agents. Research grant support is sought (a) to complete the X-ray structure determination and refinement of tomatinase, a saponin-detoxifying enzyme from Septoria lycopersici, and to pursue the structure determination of (b) related enzymes from fungi and bacteria and (c) complexes of enzymes and their mutants with substrates and inhibitors.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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