Award details

Application of combinatorial chemistry to the development of telomerase inhibitors

ReferenceB08044
Principal Investigator / Supervisor Professor Sir Shankar Balasubramanian
Co-Investigators /
Co-Supervisors
Institution University of Cambridge
DepartmentChemistry
Funding typeResearch
Value (£) 171,579
StatusCompleted
TypeResearch Grant
Start date 04/08/1997
End date 04/02/2001
Duration42 months

Abstract

The proposal aims to develop bis-specific inhibitors that are highly selective for the enzyme telomerase. The inhibitors will be used as mechanistic probes and potential anticancer lead compounds. A combinatorial synthetic approach will be developed to generate peptide library derivatives of an antisense DNA or PNA oligomer targeted at the telomerase active site. Several assay possibilities will be explored to develop a high throughput screen suitable for selecting inhibitors of telomerase from the library.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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