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Synthesis of mechanism-based inhibitors and probes for inositol monophosphatase

ReferenceB07860
Principal Investigator / Supervisor Professor David Gani
Co-Investigators /
Co-Supervisors
Institution University of Birmingham
DepartmentSchool of Chemistry
Funding typeResearch
Value (£) 91,325
StatusCompleted
TypeResearch Grant
Start date 02/06/1997
End date 02/08/1999
Duration26 months

Abstract

The mechanism and structure of inositol monophosphatase, the putative target for lithium therapy, have been determined recently in our laboratory. A new range of mechanism-based inhibitors for inositol monophosphatase will be synthesised by elaboration of O6-(2'- hydroxyethyl)-cyclohexane-1,2,4,6-tetraol phosphates and cyclic phosphates using new methodologies and incorporating solid-phase techniques starting from (-)-quinic acid. The compounds will be tested and the results will be used to test our understanding and to design and prepare highly specific compounds of potential medicinal value.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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