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Directed combinatorial chemistry - the utility of inverted libraries

ReferenceB04846
Principal Investigator / Supervisor Professor Mark Bradley
Co-Investigators /
Co-Supervisors
Institution University of Southampton
DepartmentSch of Chemistry
Funding typeResearch
Value (£) 212,031
StatusCompleted
TypeResearch Grant
Start date 01/11/1995
End date 31/10/1999
Duration48 months

Abstract

The research proposal describes a new synthetic method that allows the synthesis and inversion of fully protected combinatorial libraries followed by their C-terminal modification. We propose to utilise these inverted and modified libraries in a variety of novel applications. This includes the preparation of the first combinatorial library to contain an active site directed inhibitor, a unique and exceptionally attractive antibacterial delivery system and a quenched fluorescent assay system to determine the specificity of new proteases. The inverted library will also be used to screen synthetic receptors that were designed to bind carboxylates.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
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