Award details

Novel inositol triphosphate receptor agonists, antagonists and enzyme inhibitors

ReferenceB02137
Principal Investigator / Supervisor Dr Barry Potter
Co-Investigators /
Co-Supervisors
Professor Stefan Nahorski
Institution University of Bath
DepartmentPharmacy and Pharmacology
Funding typeResearch
Value (£) 124,655
StatusCompleted
TypeResearch Grant
Start date 12/09/1994
End date 12/09/1997
Duration36 months

Abstract

1. To synthesize novel inositol trisphosphate receptor agonists, partial agonists and antagonists based upon L-chiro-inositol 2,3,5-trisphosphorothioate and D- myo-inositol1,4,6-trisphosphorothioate. 2. To synthesize novel phosphate-tethered inositol trisphosphate analogues as conformationally restricted receptor ligands and enzyme inhibitors. 3. To exploit novel synthetic ligands biologically in permeabilised cultured cells and as metabolic enzyme inhibitors.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative X - not in an Initiative
Funding SchemeX – not Funded via a specific Funding Scheme
terms and conditions of use (opens in new window)
export PDF file