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RNA aptamers based on L-ribose as inhibitors of fibrillogenesis

Reference9810660
Principal Investigator / Supervisor Professor Peter Stockley
Co-Investigators /
Co-Supervisors
Institution University of Leeds
DepartmentInst of Molecular & Cellular Biology
Funding typeResearch
Value (£) 100,696
StatusCompleted
TypeResearch Grant
Start date 12/04/1999
End date 12/04/2001
Duration24 months

Abstract

We propose to isolate RNA aptamers which inhibit aggregate formation of the beta- amyloid peptide (1-42). Such aptamers would have potential as lead compounds in treatment for Alzheimer's patients. However, whilst aptamers with high affinity for the target are extremely likely to be isolated, the instability of RNA molecules in biological media will prevent their effective clinical use. To overcome this problem we intend to take advantage of the natural chirality of biological macromolecules to isolate tight binding aptamers, based on the non-natural enantiomer, L-ribose, which will be stable in biological fluids. Further refinement of these molecules will then be possible using nucleotide functional group variants.

Summary

unavailable
Committee Closed Committee - Biomolecular Sciences (BMS)
Research TopicsX – not assigned to a current Research Topic
Research PriorityX – Research Priority information not available
Research Initiative ROPA 1998 (ROPA1998) [1998]
Funding SchemeX – not Funded via a specific Funding Scheme
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